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Anticancer inhibitors Imatinib powder CAS 152459-95-5

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  • Imatinib | CAS 152459-95-5 | SCBT - Santa Cruz

    Imatinib, CAS: 152459-95-5, is an inhibitor of multiple tyrosine kinases. MF: C29H31N7O, MW: 493.60. Cited in 22 publications

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  • CAS No. 152459-95-5 | Sigma-Aldrich

    Imatinib for system suitability. 1 Product Result. | Match Criteria: CAS Number, Related Cas Number. Synonym: 4- [ (4-Methyl-1-piperazinyl)methyl]-N- [4-methyl-3- [ [4- (3-pyridinyl)-2-pyrimidinyl]amino] …

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  • Imatinib (STI571) | CAS 152459-95-5 | AbMole

    Imatinib (STI571) | CAS 152459-95-5 | AbMole BioScience | Imatinib Price. Imatinib is a multi-target inhibitor of v-Abl, c-Kit and PDGFR with IC50 of 0.6 μM, 0.1 μM and 0.1 μM, respectively. Buy c-Kit inhibitor Imatinib (STI571) from AbMole BioScience.

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  • Imatinib 152459-95-5 | TCI AMERICA

    Imatinib is a synthetic tyrosine (Tyr) kinase inhibitor and a molecular-targeted agent that specifically target several protein tyrosine kinases, such as stem-cell factor receptor (c-KIT), platelet-derived growth factor receptor (PDGF-R), and notably Bcr-Abl. Imatinib mesylate is used in the treatment of chronic myeloid leukemia (CML), gastrointestinal stromal tumors (GISTs) and a number of other malignancies. (The …

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  • Imatinib free base | STI571 | CAS#220127-57-1 |

    Imatinib is a synthetic tyrosine (Tyr) kinase inhibitor and a molecular-targeted agent that specifically target several protein tyrosine kinases, such as stem-cell factor receptor (c-KIT), platelet-derived growth factor receptor (PDGF-R), and notably Bcr-Abl. Imatinib

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  • Imatinib (STI571) | ≥99%(HPLC) | Selleck | PDGFR

    2021-1-22 · CAS NO. 152459-95-5 Imatinib (Gleevec)是一种多靶点酪氨酸激酶抑制剂,抑制v-Abl、c-Kit和PDGFR的IC50分别为0.6,0.1和0.1 μM。 库存: 现货

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  • Imatinib | PDGFR inhibitor | Buy Gleevec from Supplier

    CAS#: 152459-95-5 (free base) Description: Imatinib is a tyrosine kinase inhibitor with antineoplastic activity. Imatinib binds to an intracellular pocket located within tyrosine kinases (TK), thereby inhibiting ATP binding and preventing phosphorylation and the subsequent activation of growth receptors and their downstream signal transduction pathways.

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  • Imatinib (STI571) | Bcr-Abl Inhibitor | MedChemExpress

    600 行 · Imatinib (STI571, CGP057148B, Gleevec) is a multi-target inhibitor of tyrosine kinase with …

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  • 2014 « New Drug Approvals « Page 17

    Imatinib (STI571) 是一种口服生物可用的酪氨酸激酶抑制剂,可选择性抑制 BCR/ABL,v-Abl,PDGFR,c-kit 激酶活性。Imatinib (STI571) 靠近 ATP 结合位点结合,将其锁定在封闭或自我抑制的构象中,因此半竞争性抑制蛋白质的酶活性。Imatinib 还抑制 SARS-CoV ...

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  • www2.sibcb.ac.cn

    2020-2-24 · 152459-95-5 S2471 65-29-2 S2469 79660-72-3 S2468 43210-67-9 S2462 120011-70-3 S2481 89226-50-6 Loperamide hydrochloride ... Zolinza, MK-0683 is an HDAC inhibitor. Vorinostat CAS No 149647-78-9 with purity >99% & solubility DMSO is available. Vandetanib is a VEGFR and EGFR antagonist and a tyrosine kinase inhibitor with IC50 of 60, 90, 40 nM for ...

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  • API Active Pharmaceutical Ingredients - Fexofenadine ...

    2019-2-22 · Imatinib (STI571) mesylate is very effective (in vitro IC50 of 25 nM) against the chronic myeloid leukemia-causing kinase Bcr-Abl. Imatinib also efficiently inhibits Kit (in vitro IC50, 410 nM) and PDGFR (in vitro IC50, 380 nM)[2]. Imatinib (STI571) mesylate is a multi-target inhibitor of v-Abl, c-Kit and inhibits Bcr/Abl, v-Ab

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  • www.apolo.com.tw

    cas# 83480-29-9 api Voglibose is a valiolamine derivative and inhibitor of alpha-glucosidase with antihyperglycemic activity. Voglibose binds to and inhibits alpha-glucosidase, an enteric enzyme found in the brush border of the small intestines that hydrolyzes oligosaccharides and disaccharides into glucose and other monosaccharides.

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  • APExBIO

    2020-2-24 · WYE-354 is a mTOR inhibitor with an IC50 of 5 nM. Rapamycin also known as Sirolimus & Rapamune is a mTOR inhibitor. Rapamycin Sirolimus inhibits cell motility by suppression of mTOR-mediated pathways. Everolimus RAD001 also known as SDZ-RAD, Certican, Zortress, Afinitorm is TOR inhibitor available at Selleck with IC50 of 0.63 nM.

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  • Medicine by Alexandros G. Sfakianakis,Αλέξανδρος Γ ...

    2021-3-1 · ≥21.5 mg/mL in DMSO, <2.81 mg/mL in EtOH, ≥83.2 mg/mL in H2O with gentle warming ≥15.45 mg/mL in DMSO, ≥5.92 mg/mL in EtOH with ultrasonic and warming, <2.03 mg/mL in H2O ≥25.95 mg/mL in DMSO, ≥8.75 mg/mL in EtOH with ultrasonic and warming, <2.91 mg/mL in H2O ≥25.05 mg/mL in DMSO, <1.63 mg/mL in H2O

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  • Pharmaceutical co-crystal compositions - University of ...

    2020-9-17 · 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24. 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24. 1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 ...

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  • ACS Publications: Chemistry journals, books, and ...

    2019-5-25 · 3.5 3.5 3.5 3.5 1 0 250.625 57.5 20 8.125 402.75 0 0 1.6722200000000001E-3 0 0.50294099999999997 89.38 2.2028999999999999E-4 2.2028600000000001E-3 2.2024200000000001E-2 0.219806 2.1554199999999999 18.052299999999999 68.778300000000002

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  • MedChemExpress (MCE): Inhibitors, Agonists & Screening ...

    CAS Number Pathway Alternative_Names Biological Description ... TA-01 inhibitors inhibit cardiac development when applied at 5 μM. 351.3246 C20H12F3N3 C04 ... Efavirenz is a potent inhibitor of the wild-type HIV-1 RT (Ki = 2.93 nM) and exhibited a 95% inhibitory concentration of 1.5 nM for the inhibition of HIV-1 replicative spread in cell ...

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  • www2.sibcb.ac.cn

    2019-2-22 · Imatinib (STI571) mesylate is very effective (in vitro IC50 of 25 nM) against the chronic myeloid leukemia-causing kinase Bcr-Abl. Imatinib also efficiently inhibits Kit (in vitro IC50, 410 nM) and PDGFR (in vitro IC50, 380 nM)[2]. Imatinib (STI571) mesylate is a multi-target inhibitor of v-Abl, c-Kit and inhibits Bcr/Abl, v-Ab

    Get Price
  • WO 2006/135479 A2 - Anti-scarring Agents,

    Additional exemplary cyclin dependent protein kinase inhibitors include an anticancer agent from Astex Technology, a CAK1 inhibitor from GPC Biotech, a CDK inhibitor from Sanofi-Aventis, a CDK1/CDK2 inhibitor from Amgen, a CDK2 inhibitor from SUGEN-2 (Pfizer), a hearing loss therapy agent (Sound Pharmaceuticals), PD-0332991 (Pfizer), RGB-286199 ...

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  • (11) CA 2 513 746 - doczz.fr

    Commentaires . Transcription . (11) CA 2 513 746

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  • www.apexbt.com

    2021-3-1 · 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12 ...

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  • Home | Drug Metabolism & Disposition

    2018-10-12 · 95.5 3 0.98-2.2999999999999998. 1 0.38 2.3e-2 44 42 1961 284.74 3 0 32.700000000000003 1 2.8 2.8. 0.21 0.06 0.06 58 48 1961 230.67 4 1 58.5 0 1.2 1.2. 0.13 0.8 2.7 2.4 1971 451.52 13 9 247.9 6-6-8. 0.19 5.3 0.6 0.65 1885 128.94 2 1 37.299999999999997 1 0.9-2.5. 0.22 3.5 5.0000000000000001e-3 1 1.4 1968 296.14999999999998 3 2 49.3 4 4 1 ...

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  • Pharmaceutical co-crystal compositions - University of ...

    A pharmaceutical composition comprising a co-crystal of an API and a co-crystal former; wherein the API has at least one functional group selected from ether, thioether, alcohol, thiol, aldehyde, ketone, thioketone, nitrate ester, phosphate ester, thiophosphate ester, ester, thioester, sulfate ester, carboxylic acid, phosphonic acid, phosphinic acid, sulfonic acid, amide, primary amine ...

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  • Pharmaceutical propylene glycol solvate compositions ...

    Uno, T. et al. “Structure of 5,5-diphenylhydantoin-1- (4-bromophenyl)-4-dimethylamino-2,3-dimethyl-3-pyrazolin-5-one (1:1)” Acta Cryst, 1980, pp. 2794-2796, vol. B36. Van Roey, P. et al. “Structure-activity studies of non-steroidal aromatase inhibitors: the crystal and molecular structures of CGS 16949A and CGS 18320B” J. Enzyme ...

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  • WO 2006/135479 A2 - Anti-scarring Agents,

    Additional exemplary cyclin dependent protein kinase inhibitors include an anticancer agent from Astex Technology, a CAK1 inhibitor from GPC Biotech, a CDK inhibitor from Sanofi-Aventis, a CDK1/CDK2 inhibitor from Amgen, a CDK2 inhibitor from SUGEN-2 (Pfizer), a hearing loss therapy agent (Sound Pharmaceuticals), PD-0332991 (Pfizer), RGB-286199 ...

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    2021-3-1 · 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12 ...

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  • Pseudoginsenoside Rh2 | CAS:1370264-16-6 |

    2021-3-23 · ChemFaces is Reference Standard and high-purity Natural Products Manufacturer of Pseudoginsenoside Rh2(CFN93178) CAS no.:1370264-16-6

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  • Alpha Lifetech

    LY294002 is the first synthetic molecule known to inhibit PI3Kα/δ/β with IC50 of 0.5 μM/0.57 μM/0.97 μM, respectively; more stable in solution than Wortmannin, and also blocks autophagosome formation. C19H17NO3 742112-33-0 PDK-1 OSU-03012 is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM and 2-fold increase in potency over OSU ...

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  • Antiepileptic Drugs - Studyres

    Find the training resources you need for all your activities. Studyres contains millions of educational documents, questions and answers, notes about the course, tutoring questions, cards and course recommendations that will help you learn and learn.

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  • WO 2006/135479 A2 - Anti-scarring Agents,

    Additional exemplary cyclin dependent protein kinase inhibitors include an anticancer agent from Astex Technology, a CAK1 inhibitor from GPC Biotech, a CDK inhibitor from Sanofi-Aventis, a CDK1/CDK2 inhibitor from Amgen, a CDK2 inhibitor from SUGEN-2 (Pfizer), a hearing loss therapy agent (Sound Pharmaceuticals), PD-0332991 (Pfizer), RGB-286199 ...

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    2021-3-2 · 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12. 1 2 3 4 5 6 7 8 9 10 11 12 ...

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  • Alpha Lifetech

    LY294002 is the first synthetic molecule known to inhibit PI3Kα/δ/β with IC50 of 0.5 μM/0.57 μM/0.97 μM, respectively; more stable in solution than Wortmannin, and also blocks autophagosome formation. C19H17NO3 742112-33-0 PDK-1 OSU-03012 is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM and 2-fold increase in potency over OSU ...

    Get Price
  • Antiepileptic Drugs - Studyres

    Find the training resources you need for all your activities. Studyres contains millions of educational documents, questions and answers, notes about the course, tutoring questions, cards and course recommendations that will help you learn and learn.

    Get Price